SCHEMBL4539989

SCHEMBL4539989

COC(=O)c1cccn1-c1ncc(N)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
PPARG P37231 1/20 0.41
NR2E3 Q9Y5X4 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
NQO2 P16083 2/20 0.38
P2RY12 Q9H244 1/20 0.38
ALDH1A1 P00352 2/20 0.38
OPRK1 P41145 1/20 0.38
LMNA P02545 1/20 0.37
RAB9A P51151 1/20 0.36
GPX4 P36969 1/20 0.36
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4539690 0.85 MAPT (0.51) MAPTNPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL4540145 0.85 CYP1A2 (0.49) MAPTNPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL4540046 0.85 MAPT (0.43) MAPTNPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL4540292 0.82 MAPT (0.64) MAPTNPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL4539851 0.82 MAPT (0.42) MAPTNPSR1CYP3A4MEN1KMT2A
SCHEMBL4542687 0.81 MAPT (0.45) MAPTNPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL20278430 0.78 F2 (0.42) MAPTMEN1KMT2ANQO2P2RY12
SCHEMBL20265204 0.77 OPRK1 (0.39) MAPTMEN1KMT2ANQO2P2RY12
Acetonitrile SCHEMBL27922454 0.77 BDKRB1 (0.40) MAPTMEN1KMT2APPARGNR2E3
SCHEMBL28999951 0.74 ALDH1A1 (0.41) MAPTALDH1A1LMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009117421-A2 HETEROCYCLIC MODULATORS OF GPR119 FOR TREATMENT OF DISEASE KALYPSYS, INC. (US) 2009-09-24 WO disclosed