SCHEMBL4540207

SCHEMBL4540207

NC(=O)Cc1ccc(-c2ccccc2C(=O)N2CCOCC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.53
ALOX5AP P20292 1/20 0.52
FEN1 P39748 1/20 0.52
TSHR P16473 2/20 0.51
RECQL P46063 1/20 0.51
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
TP53 P04637 1/20 0.50
HTT P42858 1/20 0.48
GAA P10253 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PLAUR Q03405 1/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
FAAH O00519 1/20 0.47
MGLL Q99685 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540201 0.85 MAPT (0.51) MAPTALOX5APFEN1TSHRRECQL
SCHEMBL7885351 0.83 ALDH1A1 (0.60) MAPTALOX5APFEN1TSHRRECQL
SCHEMBL3996738 0.82 TSHR (0.73) TSHRRECQLALDH1A1CYP1A2CYP3A4
SCHEMBL31717616 0.74 PARP1 (0.59) ALDH1A1TP53HTTSMN1; SMN2
SCHEMBL22692602 0.74 PKM (0.61) TSHRALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7121916 0.74 SMN1; SMN2 (0.77) TSHRALDH1A1TP53HTTGAA
Hydrochloric Acid SCHEMBL31717432 0.73 PARP1 (0.58) ALDH1A1TP53HTTSMN1; SMN2
SCHEMBL5349455 0.73 SMN1; SMN2 (0.67) TSHRALDH1A1TP53HTTGAA
SCHEMBL15917045 0.73 ALOX5AP (0.73) ALOX5APFEN1ALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL17559454 0.72 SMN1; SMN2 (0.65) TSHRALDH1A1TP53HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed