SCHEMBL4540845

SCHEMBL4540845

CC(C)(C)OC(=O)N1CC(O)(c2c[nH]c3cc(Br)ccc23)C1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.39
ALK Q9UM73 1/20 0.38
USP30 Q70CQ3 2/20 0.37
IDO1 P14902 2/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
GSK3B P49841 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
BACE1 P56817 1/20 0.36
CYP2A6 P11509 1/20 0.36
ROCK2 O75116 1/20 0.35
PIM1 P11309 1/20 0.35
TDO2 P48775 1/20 0.35
NR4A2 P43354 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
ESR2 Q92731 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20327947 0.87 MET (0.41) RORCIDO1TDO2
SCHEMBL31530791 0.87 MET (0.41) RORCIDO1TDO2
SCHEMBL31295090 0.84 MAPT (0.44) NR4A2
SCHEMBL16610322 0.83 NR1H2 (0.36) IDO1ROCK2TDO2
SCHEMBL30053594 0.80 ALDH1A1 (0.44) RORCIDO1
SCHEMBL29206537 0.80 ALDH1A1 (0.44) RORCIDO1
SCHEMBL20530087 0.79 ALK (0.43) RORCALKIDO1BACE1TDO2
SCHEMBL31735017 0.78 RORC (0.42) RORCUSP30BACE1ROCK2ESR2
SCHEMBL25337397 0.77 BACE1 (0.50) ALKBACE1
SCHEMBL4566022 0.76 SLC6A4 (0.46) RORCUSP30IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009120655-A1 INDOLE DERIVATIVES H. LUNDBECK A/S (DK) 2009-10-01 WO disclosed