SCHEMBL4543121

SCHEMBL4543121

Cn1c(CCCCN2CCc3ccc(C#N)cc3C2)nnc1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 12/20 0.57
DRD3 P35462 11/20 0.57
DRD4 P21917 2/20 0.47
OPRM1 P35372 2/20 0.47
KCNH2 Q12809 2/20 0.46
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42
HTR7 P34969 1/20 0.42
HRH1 P35367 1/20 0.42
HTR2B P41595 1/20 0.42
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7201980 0.99 DRD2 (0.56) DRD2DRD3DRD4OPRM1KCNH2
SCHEMBL4389062 0.83 DRD3 (0.63) DRD2DRD3DRD4KCNH2HTR1A
SCHEMBL4395639 0.81 HTR7 (0.43) DRD2DRD3KCNH2HTR1AHTR2A
SCHEMBL4381610 0.78 KDM4E (0.44) DRD2DRD3KCNH2HTR7HTR2B
SCHEMBL4392739 0.77 HTT (0.42) DRD2DRD3KCNH2
SCHEMBL4766034 0.77 DRD3 (0.70) DRD2DRD3DRD4KCNH2HTR1A
Hydrochloric Acid SCHEMBL7199896 0.76 HTT (0.41) DRD2DRD3KCNH2
SCHEMBL3348927 0.74 DRD2 (1.00) DRD2DRD3DRD4OPRM1HTR1A
SCHEMBL7844061 0.73 DRD2 (0.74) DRD2DRD3DRD4OPRM1HTR1A
SCHEMBL6979746 0.70 DRD3 (0.74) DRD2DRD3DRD4OPRM1HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP disclosed