SCHEMBL454917

SCHEMBL454917

COCCc1nc(-c2cc(F)cc(F)c2)[nH]c(=O)c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNKS O95271 3/20 0.41
PARP1 P09874 3/20 0.41
TNKS2 Q9H2K2 3/20 0.41
HCAR2 Q8TDS4 1/20 0.39
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GRK6 P43250 1/20 0.35
MAPT P10636 1/20 0.35
MTOR P42345 1/20 0.35
POLB P06746 1/20 0.34
SLC9A1 P19634 1/20 0.34
PIN1 Q13526 1/20 0.34
SMPD3 Q9NY59 1/20 0.34
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL454863 0.79 WNT3A (0.39) TNKS2SMN1; SMN2DHODH
SCHEMBL19366154 0.65 PIN1 (0.49) HCAR2GRK6SLC9A1PIN1SMPD3
SCHEMBL12487639 0.65 SMN1; SMN2 (0.47) TNKSPARP1TNKS2SMN1; SMN2MAPT
SCHEMBL377866 0.60 BRD4 (0.45) TNKSPARP1TNKS2
SCHEMBL13736743 0.60 CYP1A2 (0.49) GRIN1GRIN2BSMN1; SMN2
SCHEMBL15570393 0.60 HCAR2 (0.40) HCAR2MAPTPOLB
SCHEMBL13733863 0.59 CYP1A2 (0.43) GRIN1GRIN2BSMN1; SMN2
SCHEMBL25347352 0.58 HTT (0.38) HCAR2DHODH
SCHEMBL9895127 0.58 CYP1A2 (0.47) GRIN1GRIN2BSMN1; SMN2
SCHEMBL21964587 0.57 HCAR2 (0.38) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2475654-A1 HERBICIDAL PYRIMIDONE DERIVATIVES E. I. du Pont de Nemours and Company (US) 2012-07-18 EP disclosed
WO-2012033548-A2 HERBICIDAL BIS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-15 WO disclosed
WO-2011031658-A1 HERBICIDAL PYRIMIDONE DERIVATIVES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-03-17 WO disclosed