SCHEMBL4552845

SCHEMBL4552845

O=c1ccnc(C(F)C(F)F)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.38
LMNA P02545 1/20 0.38
GPR84 Q9NQS5 1/20 0.36
PDE3B Q13370 10/20 0.35
PDE3A Q14432 10/20 0.35
L3MBTL1 Q9Y468 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
MAPT P10636 2/20 0.32
APEX1 P27695 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
DCTPP1 Q9H773 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2625456 0.75 GSK3B (0.46) POLBLMNAGPR84PDE3BPDE3A
SCHEMBL22275400 0.72 PDE3B (0.39) POLBLMNAGPR84PDE3BPDE3A
SCHEMBL6587174 0.72 PDE3B (0.42) POLBLMNAGPR84PDE3BPDE3A
Hydrochloric Acid SCHEMBL6293153 0.71 PDE3B (0.41) POLBLMNAGPR84PDE3BPDE3A
Hydrochloric Acid SCHEMBL6293152 0.71 PDE3B (0.41) POLBLMNAGPR84PDE3BPDE3A
SCHEMBL6215876 0.67
SCHEMBL3855002 0.67 HCAR2 (0.42) POLBLMNAGPR84PDE3BPDE3A
SCHEMBL22487895 0.66 GPR84 (0.44) POLBLMNAGPR84PDE3BPDE3A
SCHEMBL6293377 0.65 PDE3B (0.39) POLBLMNAGPR84PDE3BPDE3A
SCHEMBL6293376 0.65 PDE3B (0.39) POLBLMNAGPR84PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397351-B1 PYRIMIDINE, TRIAZINE AND PYRAZINE DERIVATIVES AS GLUTAMATE RECEPTORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP disclosed
CN-1146455-C 1,2,4,5-tetrahydro-benzo[d] azepine compound - 2004-04-21 CN disclosed
CN-1283623-A 1,2,4,5-tetrahydro-benzo[d] azepine compound HAFMAN RAROCHE S A F (CH) 2001-02-14 CN disclosed