SCHEMBL4553306

SCHEMBL4553306

CCN1CCC(Oc2ccc(-c3cccc([AsH2])n3)c(OC)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 7/20 0.49
HRH3 Q9Y5N1 4/20 0.43
FGFR1 P11362 2/20 0.39
PDGFRA P16234 1/20 0.39
FLT1 P17948 1/20 0.39
KDR P35968 1/20 0.39
CRHR1 P34998 1/20 0.37
KCNH2 Q12809 1/20 0.37
TTK P33981 2/20 0.37
IGF1R P08069 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
ROCK2 O75116 1/20 0.36
CCR2 P41597 1/20 0.36
ROCK1 Q13464 1/20 0.36
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL220335 0.88 CHEK1 (0.47) CHEK1HRH3FGFR1PDGFRAFLT1
SCHEMBL16241883 0.84 NOS1 (0.51) CHEK1HRH3FGFR1TTKIGF1R
SCHEMBL16241884 0.83 CHEK1 (0.48) CHEK1HRH3FGFR1TTKIGF1R
SCHEMBL221859 0.75 NOS1 (0.57) CHEK1TTKIGF1RDYRK1BROCK2
SCHEMBL221344 0.72 NOS1 (0.65) CHEK1TTKIGF1RDYRK1B
SCHEMBL5824113 0.72 PDE7A (0.49) CHEK1ROCK1
SCHEMBL221708 0.71 NOS1 (0.45) HRH3
SCHEMBL5140699 0.70 NOS3 (0.53) CHEK1TTKIGF1RDYRK1B
SCHEMBL221586 0.70 NMT1 (0.45) CHEK1KCNH2ROCK1
SCHEMBL28813994 0.69 CHEK1 (0.44) CHEK1HRH3TTKIGF1RDYRK1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158646-A1 THERAPEUTIC COMPUNDS AND RELATED METHODS OF USE ELIXIR PHARMACEUTICALS, INC. (US) 2009-12-30 WO disclosed