SCHEMBL5140699

SCHEMBL5140699

COc1cc(OC2CCN(C)C2)ccc1-c1cccc(-c2ccccc2N)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.53
NOS1 P29475 1/20 0.53
NOS2 P35228 1/20 0.53
CHEK1 O14757 3/20 0.43
USP2 O75604 1/20 0.42
USP1 O94782 1/20 0.42
USP8 P40818 1/20 0.42
OTUB1 Q96FW1 1/20 0.42
TTK P33981 2/20 0.42
PDE3B Q13370 4/20 0.41
PDE3A Q14432 4/20 0.41
PDE10A Q9Y233 4/20 0.41
IGF1R P08069 2/20 0.41
INSR P06213 1/20 0.41
ALK Q9UM73 1/20 0.41
DYRK1B Q9Y463 1/20 0.39
HTR1A P08908 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL221344 0.89 NOS1 (0.65) NOS3NOS1NOS2CHEK1TTK
SCHEMBL5134246 0.83 NMT1 (0.43) CHEK1IGF1R
SCHEMBL221859 0.83 NOS1 (0.57) NOS3NOS1NOS2CHEK1TTK
SCHEMBL5140700 0.81 CHEK1 (0.47) NOS3NOS1NOS2CHEK1TTK
SCHEMBL424370 0.81 NOS1 (0.54) NOS3NOS1NOS2CHEK1
SCHEMBL27981858 0.78 CHEK1 (0.45) NOS3NOS1NOS2CHEK1PDE3B
SCHEMBL1912083 0.77 ALDH1A1 (0.50) CHEK1PDE3BPDE3APDE10AHTR2C
SCHEMBL10208091 0.77 ALDH1A1 (0.50) CHEK1PDE3BPDE3APDE10AHTR2C
SCHEMBL1782598 0.77 ALDH1A1 (0.50) CHEK1PDE3BPDE3APDE10AHTR2C
SCHEMBL16241883 0.77 NOS1 (0.51) NOS3NOS1NOS2CHEK1TTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877054-A2 NICOTINAMIDE RIBOSIDE AND ANALOGUES THEREOF Sirtris Pharmaceuticals, Inc. (US) 2008-01-16 EP disclosed
WO-2006105440-A2 NICOTINAMIDE RIBOSIDE AND ANALOGUES THEREOF SIRTRIS PHARMACEUTICALS, INC. (US) 2006-10-05 WO disclosed