SCHEMBL4553620

SCHEMBL4553620

COC(=O)c1cccc(OC)c1OC(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
GAA P10253 2/20 0.50
KDM4E B2RXH2 2/20 0.50
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
TSHR P16473 2/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
SLC6A3 Q01959 2/20 0.43
NR1I2 O75469 1/20 0.43
CNR2 P34972 1/20 0.43
STAT3 P40763 1/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 2/20 0.42
SLC6A4 P31645 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methyl 2,3-Dimethoxybenzoate SCHEMBL311487 0.83 GAA (0.66) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL12569625 0.83 NR4A2 (0.44) ALDH1A1KDM4EPOLBKMT2ATSHR
SCHEMBL1438636 0.83 ALDH1A1 (0.59) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL12492132 0.83 ALDH1A1 (0.47) ALDH1A1KDM4EPOLBKMT2ATSHR
SCHEMBL1438500 0.81 TSHR (0.42) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL1856862 0.80 SLC6A3 (0.56) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL12545932 0.80 KDM4E (0.45) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL28000332 0.79 SMN1; SMN2 (0.48) ALDH1A1GAAKDM4ETSHRMAPT
SCHEMBL31388963 0.78 NR1I2 (0.46) ALDH1A1GAAKDM4EPOLBTSHR
SCHEMBL22726546 0.78 CA12 (0.50) ALDH1A1POLBKMT2AMAPTNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed