SCHEMBL4555697

SCHEMBL4555697

O=C1O[C@H](CO)CN1c1ccc(N2CCC3(CC2)Oc2cccc(F)c2O3)nc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CALML3 P27482 6/20 0.45
MAOA P21397 4/20 0.41
MAOB P27338 3/20 0.41
F10 P00742 1/20 0.40
CYP2C19 P33261 2/20 0.39
CYP2C9 P11712 1/20 0.39
CYP3A4 P08684 1/20 0.37
FFAR4 Q5NUL3 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
GRM2 Q14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14261417 0.77 CALML3 (0.52) CALML3MAOAMAOBF10CYP2C19
SCHEMBL14261644 0.77 CALML3 (0.52) CALML3MAOAMAOBF10CYP2C19
SCHEMBL4728137 0.75 CALML3 (0.45) CALML3MAOAMAOBF10CYP2C19
SCHEMBL14261642 0.73 CALML3 (0.43) CALML3MAOAMAOBF10CYP2C19
SCHEMBL4727825 0.73 CALML3 (0.43) CALML3MAOAMAOBF10CYP2C19
SCHEMBL14261606 0.72 F10 (0.47) CALML3MAOAMAOBF10CYP2C19
SCHEMBL4778998 0.72 F10 (0.44) CALML3MAOAMAOBF10CYP2C19
SCHEMBL4783429 0.72 F10 (0.44) CALML3MAOAMAOBF10CYP2C19
SCHEMBL14261619 0.72 PKM (0.56) CALML3MAOAMAOBF10CYP2C19
SCHEMBL4728850 0.72 PKM (0.56) CALML3MAOAMAOBF10CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037542-A2 SPIROCYCLIC COMPOUNDS AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS, S.A. (US) 2009-03-26 WO claimed