SCHEMBL4728850

SCHEMBL4728850

O=C1O[C@@H](CO)CN1c1ccc(N2CCN(S(=O)(=O)c3ccc(F)cc3F)CC2)nc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.56
CALML3 P27482 6/20 0.48
POLB P06746 1/20 0.45
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
MAOA P21397 3/20 0.44
MAOB P27338 3/20 0.44
F10 P00742 3/20 0.43
CYP3A4 P08684 1/20 0.42
PKLR P30613 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14261619 1.00 PKM (0.56) PKMCALML3POLBCYP2C19CYP2C9
SCHEMBL4728524 0.82 CNR1 (0.46) CALML3POLBMAOAMAOBF10
SCHEMBL14261644 0.79 CALML3 (0.52) CALML3CYP2C19CYP2C9MAOAMAOB
SCHEMBL14261417 0.79 CALML3 (0.52) CALML3CYP2C19CYP2C9MAOAMAOB
SCHEMBL14261606 0.77 F10 (0.47) CALML3CYP2C19CYP2C9MAOAMAOB
SCHEMBL4728137 0.75 CALML3 (0.45) CALML3CYP2C19CYP2C9MAOAMAOB
SCHEMBL4783498 0.73 KDM4E (0.49) CALML3CYP2C19CYP2C9MAOAMAOB
SCHEMBL14261404 0.73 KDM4E (0.49) CALML3CYP2C19CYP2C9MAOAMAOB
SCHEMBL10151464 0.73 MAOA (0.45) CALML3MAOAMAOBF10
SCHEMBL14261333 0.73 DDB1 (0.49) MAOAMAOBF10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008029266-A1 STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (US) 2008-03-13 WO claimed
WO-2008029266-A1 STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (US) 2008-03-13 WO disclosed