SCHEMBL4556581

SCHEMBL4556581

COC(=O)C1(O)CNC1.OC1CN(C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 5/20 0.44
CYP2D6 P10635 5/20 0.43
CYP2C9 P11712 4/20 0.43
CYP3A4 P08684 4/20 0.43
NPSR1 Q6W5P4 1/20 0.42
GPR55 Q9Y2T6 1/20 0.42
CYP2C19 P33261 3/20 0.42
CYP1A2 P05177 2/20 0.39
TSHR P16473 2/20 0.39
OPRL1 P41146 3/20 0.39
OPRM1 P35372 2/20 0.39
ACHE P22303 1/20 0.39
HIF1A Q16665 1/20 0.38
SLC6A9 P48067 1/20 0.38
OPRK1 P41145 1/20 0.38
KMT2A Q03164 1/20 0.38
USP2 O75604 1/20 0.38
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1602301 0.77 CYP3A4 (0.57) OPRD1CYP2D6CYP2C9CYP3A4NPSR1
SCHEMBL48800 0.75 OPRM1 (0.48) OPRD1CYP2D6OPRL1OPRM1SLC6A9
SCHEMBL5745379 0.74 CYP2D6 (0.47) OPRD1CYP2D6CYP2C9CYP3A4CYP2C19
Hydrochloric Acid SCHEMBL741583 0.73 OPRM1 (0.47) OPRD1CYP2D6OPRL1OPRM1SLC6A9
SCHEMBL19281773 0.73 OPRM1 (0.47) OPRD1CYP2D6OPRL1OPRM1SLC6A9
SCHEMBL72964 0.70 CYP3A4 (0.49) OPRD1CYP2D6CYP2C9CYP3A4CYP2C19
SCHEMBL1603102 0.70
Hydrochloric Acid SCHEMBL5198335 0.70 OPRM1 (0.41) OPRD1CYP2D6OPRL1OPRM1ACHE
SCHEMBL20133104 0.70 OPRM1 (0.54) OPRD1CYP2D6OPRL1OPRM1SLC6A9
SCHEMBL6011821 0.69 OPRD1 (0.57) OPRD1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP disclosed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed