SCHEMBL4556840

SCHEMBL4556840

O=C(c1ccc(Cn2c(C(F)(F)F)nc3ccccc32)cc1)C(O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.55
CYP2C19 P33261 3/20 0.55
CYP1A2 P05177 2/20 0.55
CYP2D6 P10635 1/20 0.55
CYP3A4 P08684 1/20 0.52
PPARG P37231 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
ADAMTS4 O75173 1/20 0.49
MMP12 P39900 1/20 0.49
ADAM17 P78536 1/20 0.49
ADAMTS5 Q9UNA0 1/20 0.49
LMNA P02545 3/20 0.47
TSHR P16473 1/20 0.47
TP53 P04637 1/20 0.47
AGTR1 P30556 2/20 0.46
AGTR2 P50052 2/20 0.46
ALDH1A1 P00352 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HDAC1 Q13547 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4556839 0.96 CYP2C9 (0.58) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL4048200 0.85 CYP2C9 (0.63) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL14376771 0.80 HDAC1 (0.69) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL23430141 0.78 TNF (0.49) CYP2C9CYP2C19CYP1A2CYP2D6MEN1
SCHEMBL24041745 0.77 CYP2C9 (0.54) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL13508742 0.76 NOD1 (0.62) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL6244545 0.76 AGTR1 (0.65) CYP2C9CYP2C19CYP1A2PPARGMEN1
SCHEMBL28388694 0.75 TNF (0.54) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL4445288 0.74 CYP2C9 (0.51) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4
SCHEMBL4445291 0.74 CYP2C9 (0.51) CYP2C9CYP2C19CYP1A2CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397137-B1 HYDANTION DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES BRISTOL MYERS SQUIBB CO (US) 2009-10-14 EP disclosed