SCHEMBL4558101

SCHEMBL4558101

CCC(=O)Nc1ccc2c(c1)C(C)(C)C(C)=N2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.48
CYP3A4 P08684 3/20 0.47
TSHR P16473 1/20 0.43
POLB P06746 3/20 0.43
NR4A1 P22736 1/20 0.43
BACE1 P56817 1/20 0.43
CASP3 P42574 1/20 0.43
GAA P10253 3/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27142760 0.85 KMT2A (0.37) RAB9ACYP3A4POLBALDH1A1MAPT
SCHEMBL4506249 0.84 MEN1 (0.45) RAB9ACYP3A4TSHRPOLBBACE1
SCHEMBL25083574 0.83 BRAF (0.34) RAB9ACYP3A4POLBBACE1MAPT
SCHEMBL12496810 0.80 TDP1 (0.44) RAB9APOLBGAAALDH1A1MAPT
SCHEMBL11234029 0.78 NPC1 (0.52) RAB9ACYP3A4POLBGAAMAPT
SCHEMBL4502019 0.76 MEN1 (0.37) MEN1KMT2APDK2
SCHEMBL917056 0.70 POLB (0.54) RAB9ACYP3A4TSHRPOLBNR4A1
SCHEMBL5695447 0.70 TDP1 (0.39) RAB9ACASP3GAAALDH1A1MAPT
SCHEMBL11734764 0.70 ALDH1A1 (0.44) RAB9ACYP3A4POLBGAAALDH1A1
SCHEMBL8390740 0.70 CA2 (0.40) RAB9ACYP3A4POLBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592188-B2 environmentally sensitive fluorescent dye covalently linked to a binding domain which has specific affinity for a target molecule; fluorescence resonance energy transfer; detecting changes in the binding, conformational change; detecting human immunodeficiency virus THE SCRIPPS RESEARCH INSTITUTE (US) 2009-09-22 US disclosed
US-20060029946-A1 Live cell biosensors NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2006-02-09 US disclosed