SCHEMBL4558326

SCHEMBL4558326

CC(C)C(N)C(=O)OCn1ccnn1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.36
CYP19A1 P11511 12/20 0.36
CYP1A1 P04798 2/20 0.36
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK1 P28482 1/20 0.32
HBB P68871 1/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
DPP4 P27487 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27739344 0.73 ALDH1A1 (0.44) FOLH1CYP19A1CYP1A1
SCHEMBL19941705 0.73 THRB (0.41) MEN1KMT2AMAPK1HBBHSP90AA1
SCHEMBL21990274 0.72 FOLH1 (0.36) FOLH1CYP19A1CYP1A1KMT2A
SCHEMBL28807834 0.72 FOLH1 (0.39) FOLH1CYP19A1CYP1A1
SCHEMBL7259407 0.69 CYP19A1 (0.38) FOLH1CYP19A1
SCHEMBL29201284 0.67 CYP19A1 (0.48) FOLH1CYP19A1CYP1A1
SCHEMBL28468849 0.67 CYP19A1 (0.48) FOLH1CYP19A1CYP1A1
SCHEMBL21722399 0.67 CYP19A1 (0.48) FOLH1CYP19A1CYP1A1
SCHEMBL9284133 0.67 CYP19A1 (0.58) CYP19A1CYP1A1KMT2AMAPK1
SCHEMBL22551813 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035396-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-03-18 EP disclosed
WO-2007139967-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO disclosed