SCHEMBL4558438

SCHEMBL4558438

CCc1c2ccc(-c3ccnn3-c3ccc(S(N)(=O)=O)cc3)cc2nn1C.CCc1nn(C)c2cc(-c3ccnn3-c3ccc(C#N)cc3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 5/20 0.43
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
PTGS2 P35354 10/20 0.42
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
PTGS1 P23219 3/20 0.35
CA12 O43570 3/20 0.35
CHRNA7 P36544 2/20 0.33
CYP11B2 P19099 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3599265 0.87 PTGS2 (0.44) CA9CA1CA2PTGS2PTGS1
SCHEMBL3615539 0.87 PTGS2 (0.44) CA9CA1CA2PTGS2PTGS1
SCHEMBL3612595 0.84 CYP11B2 (0.44) CA9CA1CA2CYP11B2
SCHEMBL3606471 0.84 KHK (0.40) CA9CA1CA2CYP11B2
SCHEMBL3608038 0.79 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL3602376 0.79 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL4558167 0.78 KDM5A (0.45) CA9PTGS2CA12CHRNA7
SCHEMBL8268988 0.75 KHK (0.41)
SCHEMBL8268992 0.75 MAPK9 (0.36) PTGS2
SCHEMBL3612178 0.73 PTGS2 (0.39) CA9CA1CA2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067607-A2 COMBINATIONS OF PDE4 INHIBITORS AND ANTIPSYCHOTICS FOR THE TREATMENT OF PSYCHOTIC DISORDERS MEMORY PHARMACEUTICALS CORPORATION (US) 2009-05-28 WO disclosed