SCHEMBL8268992

SCHEMBL8268992

CCc1c2ccc(-c3ccnn3-c3ccc(N)cc3)cc2nn1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK9 P45984 2/20 0.36
MAPK10 P53779 2/20 0.36
MAPK8 P45983 1/20 0.36
NR3C2 P08235 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PI4KA P42356 1/20 0.34
PIK3CG P48736 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
MAPK14 Q16539 3/20 0.34
ALDH1A1 P00352 1/20 0.33
NT5E P21589 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3612595 0.87 CYP11B2 (0.44) MAPK9MAPK10MAPK8MAPK14NT5E
SCHEMBL3615539 0.86 PTGS2 (0.44) LMNATSHRMAPK14PTGS2
SCHEMBL3604665 0.85 RARG (0.42) NR3C2
SCHEMBL3608038 0.85 PTGS2 (0.41) NT5EPTGS2
SCHEMBL8268988 0.80 KHK (0.41) MAPK9MAPK10MAPK8NR3C2SMN1; SMN2
SCHEMBL4558438 0.75 CA9 (0.43) PTGS2
SCHEMBL3594691 0.71 PTGS2 (0.39) NT5EPTGS2
SCHEMBL8269687 0.70 SIGMAR1 (0.32) MAPK14PTGS2
SCHEMBL3607275 0.70 PTGS2 (0.44) NT5EPTGS2
SCHEMBL8268975 0.70 KHK (0.41) PIK3CDKHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006044528-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2006-04-27 WO disclosed