SCHEMBL4558994

SCHEMBL4558994

CC(C)(C)OC(=O)c1ccc2c(Br)cn([Si](C)(C)C(C)(C)C)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
GABRA1 P14867 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
RHEB Q15382 2/20 0.34
SRD5A1 P18405 1/20 0.33
MAP3K5 Q99683 3/20 0.32
SLC7A5 Q01650 1/20 0.32
STAT3 P40763 2/20 0.32
ABCG2 Q9UNQ0 2/20 0.32
ALOX15 P16050 1/20 0.32
NOTUM Q6P988 1/20 0.32
GABRA5 P31644 1/20 0.31
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21824161 0.73 GABRA1 (0.36) GABRG2GABRB3GABRA1GABRA3GABRA2
SCHEMBL3102877 0.72 NOTUM (0.43) CA12CA1CA2CA9CA14
SCHEMBL940060 0.71 BRD4 (0.37) LMNA
SCHEMBL22778008 0.69 HCAR3 (0.41) LMNA
SCHEMBL29714377 0.69 HCAR3 (0.41) LMNA
SCHEMBL15566143 0.68 L3MBTL1 (0.40) HSD17B10LMNA
SCHEMBL1132147 0.67 CHRNA1 (0.51) GABRG2GABRB3GABRA1GABRA3GABRA2
SCHEMBL17495245 0.67 CA12 (0.46) GABRG2GABRB3GABRA1GABRA3GABRA2
SCHEMBL2609133 0.67 CA12 (0.50) GABRG2GABRB3GABRA1GABRA3GABRA2
SCHEMBL10776576 0.67 ESR1 (0.55) GABRG2GABRB3GABRA1GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed