SCHEMBL456303

SCHEMBL456303

Ic1[c]c(I)c(-c2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.36
ALOX5 P09917 1/20 0.35
ALDH1A1 P00352 5/20 0.35
HSD17B10 Q99714 2/20 0.34
CYP2A6 P11509 2/20 0.34
HPGD P15428 1/20 0.34
BCL2L1 Q07817 1/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
PARP1 P09874 1/20 0.32
ESR2 Q92731 1/20 0.32
CTRC Q99895 2/20 0.31
DPP4 P27487 1/20 0.31
HDAC4 P56524 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
CYP2B6 P20813 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455502 0.78 BACE1 (0.33) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL457904 0.78 CYP2A6 (0.41) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL457819 0.78 ESR2 (0.38) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL456233 0.78 ESR2 (0.38) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL454501 0.74 TP53 (0.32) BACE1ALOX5ESR2DPP4
SCHEMBL3360517 0.69 ALDH1A1 (0.47) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL456035 0.68 ALDH1A1 (0.39) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL13445421 0.67 BACE1 (0.44) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL4082425 0.65 BACE1 (0.61) BACE1ALOX5ALDH1A1HSD17B10CYP2A6
SCHEMBL7803626 0.64 BACE1 (0.52) BACE1ALOX5ALDH1A1HSD17B10CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed