SCHEMBL456233

SCHEMBL456233

Cc1[c]c(I)ccc1-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.38
CYP2A6 P11509 2/20 0.36
CYP2B6 P20813 1/20 0.36
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
BACE1 P56817 1/20 0.33
ALOX5 P09917 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
ALDH1A1 P00352 4/20 0.32
HSD17B10 Q99714 2/20 0.32
HPGD P15428 1/20 0.32
BCL2L1 Q07817 1/20 0.32
MAPK1 P28482 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
PARP10 Q53GL7 1/20 0.31
PARP11 Q9NR21 1/20 0.31
HTR7 P34969 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4371389 0.78 ESR2 (0.41) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL456303 0.78 BACE1 (0.36) ESR2CYP2A6CYP2B6BACE1ALOX5
SCHEMBL27714313 0.75 ESR2 (0.47) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL456995 0.75 ALDH1A1 (0.41) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL6206554 0.75 CYP2A6 (0.41) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL28926395 0.73 BACE1 (0.44) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL457819 0.71 ESR2 (0.38) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL454919 0.71 ESR2 (0.35) ESR2CYP2A6CYP2B6AKT1AKT2
SCHEMBL5611087 0.70 KEAP1 (0.43) AKT1AKT2BACE1ALOX5ALDH1A1
SCHEMBL3145873 0.70 NAPRT (0.43) ALDH1A1HSD17B10HPGDMAPK1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed