SCHEMBL4563226

SCHEMBL4563226

CCCCCn1nccc1CC#N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 4/20 0.40
MPO P05164 3/20 0.36
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 2/20 0.34
GLA P06280 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SAE1 Q9UBE0 1/20 0.34
UBA2 Q9UBT2 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
MEN1 O00255 1/20 0.33
CRHBP P24387 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861630 0.80 SLC9A1 (0.40) SLC9A1MPOALDH1A1HPGDHSD17B10
SCHEMBL16815457 0.78 SLC9A1 (0.39) SLC9A1MPOCYP1A2CYP2C9CYP2C19
SCHEMBL10772453 0.77 SLC9A1 (0.38) SLC9A1MPOALDH1A1KDM4EGLA
SCHEMBL11499176 0.75 SLC9A1 (0.42) SLC9A1MPOALDH1A1CYP1A2CYP2C9
SCHEMBL16861288 0.75 SLC9A1 (0.37) SLC9A1MPOALDH1A1HPGDHSD17B10
SCHEMBL2494852 0.74 SLC9A1 (0.36) SLC9A1MPOALDH1A1KDM4EPOLB
SCHEMBL31287918 0.74 SLC9A1 (0.44) SLC9A1MPOALDH1A1KDM4EPOLB
SCHEMBL13500287 0.74 SLC9A1 (0.39) SLC9A1MPOALDH1A1POLBMAPT
SCHEMBL2777756 0.73
SCHEMBL4553490 0.73 MAPK1 (0.44) ALDH1A1KDM4EHPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121621-B1 LXR AND FXR MODULATORS EXELIXIS PATENT CO LLC (US) 2014-05-07 EP disclosed
EP-2121621-A1 LXR AND FXR MODULATORS Exelixis, Inc. (US) 2009-11-25 EP disclosed
WO-2008073825-A1 LXR AND FXR MODULATORS EXELIXIS, INC. (US) 2008-06-19 WO disclosed