SCHEMBL4563531

SCHEMBL4563531

CC(C)c1cc(OC2CCN(C)C2)ccc1-c1cccc(N)n1.CC(C)c1cc(Oc2ccn(C)c2)ccc1-c1cccc(N)n1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 5/20 0.53
NOS1 P29475 5/20 0.53
NOS2 P35228 5/20 0.53
SOS1 Q07889 2/20 0.36
USP2 O75604 1/20 0.35
USP1 O94782 1/20 0.35
USP8 P40818 1/20 0.35
OTUB1 Q96FW1 1/20 0.35
PRMT5 O14744 2/20 0.33
WDR77 Q9BQA1 2/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
ATM Q13315 1/20 0.33
MCHR1 Q99705 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL954571 0.90 NOS3 (0.64) NOS3NOS1NOS2SOS1USP2
SCHEMBL221052 0.90 NOS3 (0.64) NOS3NOS1NOS2SOS1USP2
SCHEMBL4563534 0.89 NOS3 (0.40) NOS3NOS1NOS2SOS1USP2
SCHEMBL220425 0.85 NOS3 (0.56) NOS3NOS1NOS2SOS1CDK2
SCHEMBL222403 0.84 NOS3 (0.54) NOS3NOS1NOS2SOS1USP2
SCHEMBL422148 0.78 NOS3 (0.47) NOS3NOS1NOS2SOS1USP2
SCHEMBL221344 0.76 NOS1 (0.65) NOS3NOS1NOS2PDE3BPDE3A
SCHEMBL6584972 0.76 NOS3 (0.62) NOS3NOS1NOS2USP2USP1
SCHEMBL956395 0.74 NOS3 (0.60) NOS3NOS1NOS2USP2USP1
SCHEMBL221743 0.73 PRKCZ (0.45) NOS3NOS1NOS2SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158646-A1 THERAPEUTIC COMPUNDS AND RELATED METHODS OF USE ELIXIR PHARMACEUTICALS, INC. (US) 2009-12-30 WO disclosed
WO-2006094210-A2 TETRAHYDROQUINOXALINONE SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2006-09-08 WO disclosed