SCHEMBL4563773

SCHEMBL4563773

Cc1cc(-c2ccccc2)c2nc(C3CCCN3C(=O)O)cn2c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
HCRTR1 O43613 13/20 0.41
HCRTR2 O43614 13/20 0.41
TRPV1 Q8NER1 1/20 0.40
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
SCD5 Q86SK9 3/20 0.38
SCD O00767 1/20 0.38
GRM5 P41594 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14145065 0.91 HCRTR1 (0.45) DRD2DRD4DRD3HCRTR1HCRTR2
SCHEMBL341458 0.86 GFER (0.47)
SCHEMBL342144 0.84 ALDH1A3 (0.50) HCRTR1HCRTR2TRPV1SCD5SCD
SCHEMBL342015 0.79 TRPV1 (0.38) HCRTR1HCRTR2TRPV1SCD5SCD
SCHEMBL343089 0.79 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL10182858 0.78 XIAP (0.43)
SCHEMBL14145066 0.77 HCRTR1 (0.40) DRD2DRD4DRD3HCRTR1HCRTR2
SCHEMBL342337 0.74 ALDH1A3 (0.40) HCRTR1HCRTR2TRPV1
SCHEMBL14144746 0.74 ALDH1A3 (0.47) HCRTR1HCRTR2SCD5SCDGRM5
SCHEMBL4563122 0.74 SCD5 (0.42) HCRTR1HCRTR2TRPV1SCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125809-A1 IMIDAZOPYRIDINE INHIBITORS OF IAP Genentech, Inc. (US) 2009-12-02 EP disclosed
WO-2008079735-A1 IMIDAZOPYRIDINE INHIBITORS OF IAP GENENTECH, INC. (US) 2008-07-03 WO disclosed