SCHEMBL4563902

SCHEMBL4563902

CC(C)C[C@H](C(=O)O)N(Cc1ccc(N)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.43
F7 P08709 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PPID Q08752 1/20 0.35
PSEN1 P49768 2/20 0.35
PSEN2 P49810 2/20 0.35
APH1B Q8WW43 2/20 0.35
NCSTN Q92542 2/20 0.35
APH1A Q96BI3 2/20 0.35
PSENEN Q9NZ42 2/20 0.35
MMP1 P03956 2/20 0.34
MMP3 P08254 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18203971 1.00 AAK1 (0.43) AAK1F7HDAC3HDAC1HDAC2
SCHEMBL18203970 1.00 AAK1 (0.43) AAK1F7HDAC3HDAC1HDAC2
SCHEMBL560617 0.88 AAK1 (0.39) AAK1F7HDAC3HDAC1HDAC2
SCHEMBL560618 0.88 AAK1 (0.39) AAK1F7HDAC3HDAC1HDAC2
SCHEMBL4564346 0.84 ALDH1A1 (0.42) HDAC3HDAC1HDAC2NCOR2ALDH1A1
SCHEMBL4564347 0.84 ALDH1A1 (0.42) HDAC3HDAC1HDAC2NCOR2ALDH1A1
SCHEMBL4445852 0.84 NR1D1 (0.44)
SCHEMBL4445860 0.84 NR1D1 (0.44)
SCHEMBL3143341 0.83 MEN1 (0.42) AAK1HDAC3HDAC1HDAC2NCOR2
SCHEMBL2544106 0.82 AAK1 (0.39) AAK1RENMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013175-A1 p38 MAP KINASE INHIBITORS Chroma Therapeutics Limited (GB) 2009-01-14 EP disclosed
WO-2007129040-A1 p38 MAP KINASE INHIBITORS CHROMA THERAPEUTICS LTD. (GB) 2007-11-15 WO disclosed