SCHEMBL4566574

SCHEMBL4566574

CC(O)c1ccc2cc(Br)c(C(F)(F)[PH](=O)O)cc2c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UGT2B7 P16662 1/20 0.43
PTPN1 P18031 8/20 0.41
PTPN2 P17706 1/20 0.36
PTPRC P08575 1/20 0.34
CYP17A1 P05093 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MMP9 P14780 1/20 0.32
PTPN5 P54829 1/20 0.31
NOTUM Q6P988 1/20 0.31
PLG P00747 1/20 0.30
PLAU P00749 1/20 0.30
AKR1C3 P42330 3/20 0.30
AKR1C2 P52895 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4414756 0.79 PTPN1 (0.67) UGT2B7PTPN1PTPN2PTPRCPTPN5
SCHEMBL4563376 0.77 PTPN1 (0.43) PTPN1PTPRC
SCHEMBL3264596 0.76 PTPN1 (0.46) PTPN1PTPN2PTPRC
SCHEMBL4566575 0.74 PTPN1 (0.44) PTPN1PTPN2PTPRC
SCHEMBL2693268 0.73 PTPN1 (0.47) UGT2B7PTPN1PTPN2PTPRCCYP17A1
SCHEMBL18300941 0.72 NOTUM (0.46) UGT2B7CYP17A1CYP2C9CYP2C19PTPN5
SCHEMBL5610446 0.69 UGT2B7 (0.82) UGT2B7CYP17A1CYP2C9CYP2C19PLG
SCHEMBL24779222 0.66 UGT2B7 (0.64) UGT2B7MMP9PLGPLAUAKR1C3
SCHEMBL30628955 0.66 UGT2B7 (0.64) UGT2B7MMP9PLGPLAUAKR1C3
SCHEMBL18562108 0.65 UGT2B7 (0.62) UGT2B7MMP9PLGPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114971-A1 FUSED AROMATIC PTP-1B INHIBITORS Merck Frosst Canada Ltd. (CA) 2009-11-11 EP disclosed
WO-2008089581-A1 FUSED AROMATIC PTP-1B INHIBITORS MERCK FROSST CANADA LTD. (CA) 2008-07-31 WO disclosed