SCHEMBL4573147

SCHEMBL4573147

COc1cc(N2CCN(C(=O)O)C(C)C2)ncc1Br

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 7/20 0.39
ROCK2 O75116 2/20 0.39
PRKG1 Q13976 2/20 0.39
SUV39H2 Q9H5I1 3/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
TACR3 P29371 2/20 0.38
RBP4 P02753 1/20 0.37
PIK3CD O00329 1/20 0.37
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
HDAC1 Q13547 1/20 0.36
PARP1 P09874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117495 0.86 HDAC1 (0.50) GRM1SUV39H2PIK3CDHDAC1
SCHEMBL4573910 0.86 HDAC1 (0.50) GRM1SUV39H2PIK3CDHDAC1
SCHEMBL4573353 0.84 CTSB (0.42) GRM1ROCK2PRKG1CTSBCTSS
SCHEMBL17310021 0.80 KDM4E (0.43) PARP1
SCHEMBL25187577 0.78 GRM1 (0.45) GRM1PIK3CDHDAC1
SCHEMBL4573090 0.77 CHRM4 (0.45) GRM1PIK3CD
SCHEMBL20210778 0.77 SUV39H2 (0.36) GRM1SUV39H2RBP4
SCHEMBL17310137 0.77 SUV39H2 (0.36) GRM1SUV39H2RBP4
SCHEMBL4574023 0.77 PIK3CD (0.43) GRM1ROCK2PRKG1PIK3CDCTSB
SCHEMBL21808506 0.77 GRM1 (0.50) GRM1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed