SCHEMBL4573353

SCHEMBL4573353

COc1cc(N2CCN(C(=O)O)C(C)C2)ncc1C1CC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.42
CTSS P25774 2/20 0.42
CTSK P43235 2/20 0.42
GRM1 Q13255 6/20 0.40
PANK3 Q9H999 4/20 0.39
TRPC6 Q9Y210 7/20 0.38
ROCK2 O75116 1/20 0.38
PRKG1 Q13976 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8107805 0.86 HDAC1 (0.49) CTSBCTSSCTSKGRM1PANK3
SCHEMBL4573147 0.84 GRM1 (0.39) CTSBCTSSCTSKGRM1ROCK2
SCHEMBL4572967 0.78 CHRM4 (0.46) GRM1
SCHEMBL4573074 0.76 CTSB (0.45) CTSBCTSSCTSKGRM1PANK3
SCHEMBL4573182 0.76 PIK3CD (0.41) CTSBCTSSCTSKGRM1
SCHEMBL8123583 0.75 ZAP70 (0.45) TRPC6
SCHEMBL4573061 0.74 ROCK2 (0.48) GRM1ROCK2PRKG1
SCHEMBL16334066 0.72 HDAC1 (0.49) GRM1ROCK2PRKG1
SCHEMBL24890694 0.71 NPC1 (0.61) GRM1
SCHEMBL4573206 0.71 PIK3CD (0.38) GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed