SCHEMBL4573317

SCHEMBL4573317

COc1cc(N2CCNCC2)ccc1C(C)(C)C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.50
HTR7 P34969 2/20 0.50
CHRNB2 P17787 2/20 0.48
CHRNA4 P43681 2/20 0.48
ADRB1 P08588 5/20 0.47
HTR3E A5X5Y0 2/20 0.47
HTR3B O95264 2/20 0.47
HTR3A P46098 2/20 0.47
HTR3D Q70Z44 2/20 0.47
HTR3C Q8WXA8 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
ALK Q9UM73 2/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
TGFBR1 P36897 3/20 0.44
ACVR1 Q04771 3/20 0.44
ACVR1B P36896 2/20 0.44
KCNH2 Q12809 1/20 0.44
DRD2 P14416 2/20 0.43
DRD3 P35462 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16001200 0.85 ADRB1 (0.53) HTR1AHTR7CHRNB2CHRNA4ADRB1
SCHEMBL8114648 0.84 CHEK1 (0.47) HTR1AHTR7ALKCHEK1
SCHEMBL4573103 0.82 ADRB1 (0.58) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL4573471 0.81 ADRB1 (0.56) HTR1AHTR7CHRNB2CHRNA4ADRB1
SCHEMBL24989042 0.78 ADRB1 (0.51) HTR1AHTR7CHRNB2CHRNA4ADRB1
SCHEMBL4573825 0.77 ACVR1 (0.51) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL361649 0.77 ADRB1 (0.61) HTR1AHTR7CHRNB2CHRNA4ADRB1
SCHEMBL22601531 0.76 ADRB1 (0.53) HTR1AHTR7CHRNB2CHRNA4ADRB1
Hydrochloric Acid SCHEMBL7711565 0.75 ADRB1 (0.59) HTR1AHTR7CHRNB2CHRNA4ADRB1
Hydrochloric Acid SCHEMBL2156292 0.75 ADRB1 (0.59) HTR1AHTR7CHRNB2CHRNA4ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed