SCHEMBL4573103

SCHEMBL4573103

Cc1cc(N2CCNCC2)ccc1C(C)(C)C#N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 9/20 0.58
DRD2 P14416 1/20 0.47
DRD3 P35462 1/20 0.47
HTR7 P34969 3/20 0.43
HTR3E A5X5Y0 5/20 0.42
HTR3B O95264 5/20 0.42
HTR3A P46098 5/20 0.42
HTR3D Q70Z44 5/20 0.42
HTR3C Q8WXA8 5/20 0.42
SIGMAR1 Q99720 5/20 0.42
HTR5A P47898 1/20 0.42
HTR1A P08908 3/20 0.42
MAPKAPK2 P49137 1/20 0.40
HTR1D P28221 2/20 0.40
HTR1B P28222 1/20 0.40
HTR2C P28335 2/20 0.39
ALDH1A1 P00352 1/20 0.39
THRB P10828 2/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573471 0.84 ADRB1 (0.56) ADRB1DRD2DRD3HTR7HTR3E
SCHEMBL14008974 0.83 ADRB1 (0.67) ADRB1HTR7HTR3EHTR3BHTR3A
SCHEMBL4573317 0.82 HTR1A (0.50) ADRB1DRD2DRD3HTR7HTR3E
SCHEMBL4573172 0.77 ADRB1 (0.53) ADRB1DRD2DRD3HTR3EHTR3B
SCHEMBL24990170 0.76 ADRB1 (0.65) ADRB1DRD2DRD3HTR7HTR3E
SCHEMBL4573342 0.75 ADRB1 (0.55) ADRB1HTR7HTR3EHTR3BHTR3A
SCHEMBL221254 0.74 ADRB1 (1.00) ADRB1HTR7HTR3EHTR3BHTR3A
SCHEMBL19579561 0.74 ADRB1 (0.67) ADRB1HTR7HTR3EHTR3BHTR3A
SCHEMBL11627069 0.73 ADRB1 (0.65) ADRB1HTR7HTR3EHTR3BHTR3A
SCHEMBL20171856 0.70 ADRB1 (0.71) ADRB1DRD2DRD3HTR7HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed