SCHEMBL4573348

SCHEMBL4573348

CC(C)(C(=O)O)c1ccc(N2CCNCC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
USP2 O75604 1/20 0.54
TSHR P16473 1/20 0.54
HSD17B10 Q99714 1/20 0.54
ADRB1 P08588 6/20 0.51
HTR3E A5X5Y0 3/20 0.50
HTR3B O95264 3/20 0.50
HTR3A P46098 3/20 0.50
HTR3D Q70Z44 3/20 0.50
HTR3C Q8WXA8 3/20 0.50
SIGMAR1 Q99720 3/20 0.50
MAOB P27338 1/20 0.48
HTR6 P50406 4/20 0.46
KDM4E B2RXH2 1/20 0.45
LMNA P02545 1/20 0.45
LTA4H P09960 1/20 0.45
SIRT6 Q8N6T7 1/20 0.45
HPGD P15428 1/20 0.44
ADRB2 P07550 1/20 0.43
NCF1 P14598 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4541552 0.86 ADRB1 (0.50) ALDH1A1USP2TSHRHSD17B10ADRB1
SCHEMBL4538749 0.83 ADRB1 (0.51) ALDH1A1USP2TSHRHSD17B10ADRB1
SCHEMBL8099474 0.83 ADRB1 (0.47) ALDH1A1USP2TSHRHSD17B10ADRB1
SCHEMBL26472636 0.82 KMT2A (0.55) ALDH1A1KDM4ELMNASIRT6
SCHEMBL12088780 0.80 ADRB1 (0.58) ALDH1A1USP2TSHRHSD17B10ADRB1
SCHEMBL20424733 0.79 KDM4E (0.59) ALDH1A1KDM4ELMNA
SCHEMBL270283 0.79 ADRB1 (0.62) ALDH1A1USP2TSHRHSD17B10ADRB1
SCHEMBL15577925 0.78 MAPT (0.52) ALDH1A1LMNA
SCHEMBL27901112 0.77 ADRB1 (0.44) ALDH1A1USP2TSHRHSD17B10ADRB1
Trifluoroacetic Acid SCHEMBL6336692 0.76 ADRB1 (0.69) ALDH1A1USP2TSHRHSD17B10ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed