SCHEMBL8099474

SCHEMBL8099474

CNC(=O)C(C)(C)c1ccc(N2CCNCC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 6/20 0.47
ALDH1A1 P00352 3/20 0.47
USP2 O75604 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MAOB P27338 1/20 0.45
HTR3E A5X5Y0 3/20 0.44
HTR3B O95264 3/20 0.44
HTR3A P46098 3/20 0.44
HTR3D Q70Z44 3/20 0.44
HTR3C Q8WXA8 3/20 0.44
SIGMAR1 Q99720 3/20 0.44
NPY2R P49146 1/20 0.43
ILK Q13418 1/20 0.43
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
MAPKAPK2 P49137 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573348 0.83 ALDH1A1 (0.54) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL4538749 0.82 ADRB1 (0.51) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL4541552 0.82 ADRB1 (0.50) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL532079 0.78 ALDH1A1 (0.59) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL4573263 0.77 MAPT (0.58) ALDH1A1TSHRNPY2RMAPTLMNA
SCHEMBL12088780 0.76 ADRB1 (0.58) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL270283 0.76 ADRB1 (0.62) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL13853439 0.73 MAPT (0.51) ADRB1ALDH1A1USP2TSHRHSD17B10
Phenylpiperazine SCHEMBL3894076 0.72 ALDH1A1 (0.63) ADRB1ALDH1A1USP2TSHRHSD17B10
SCHEMBL17675 0.71 ADRB1 (0.51) ADRB1ALDH1A1USP2TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed