SCHEMBL4574083

SCHEMBL4574083

CCOC(=O)c1cn2c(C)c(C)nc2c2c1CCC1(CCc3cc(F)ccc31)O2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
ALDH1A1 P00352 4/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 2/20 0.33
CASP3 P42574 1/20 0.33
ATM Q13315 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
GABRG2 P18507 4/20 0.33
GABRB3 P28472 4/20 0.33
GABRA5 P31644 4/20 0.33
P2RY12 Q9H244 3/20 0.33
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
NPSR1 Q6W5P4 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4573882 0.88 SMN1; SMN2 (0.34) TSHRALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4574520 0.83 SMN1; SMN2 (0.38) ALDH1A1HPGDHSD17B10SMN1; SMN2NPC1
SCHEMBL4574395 0.76 HCAR2 (0.35) ALDH1A1CYP3A4CYP2C9
SCHEMBL5323237 0.74 AKT1 (0.35) TSHRALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4575118 0.73 HCRTR1 (0.30)
SCHEMBL4597065 0.73 HCRTR1 (0.33) HPGDSMN1; SMN2LMNA
SCHEMBL4595427 0.72 LMNA (0.35) TSHRALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL4737833 0.68 BRD4 (0.31)
SCHEMBL4737642 0.67 NPY5R (0.37) TSHRALDH1A1HPGDNPC1RAB9A
SCHEMBL14068758 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008071766-A2 SPIRO-INDENE SUBSTITUTED IMIDAZONAPHYTHYRIDINE AND PYRANOIMIDAZOPYRIDINE DERIVATIVES AS INHIBITORS OF GASTRIC ACID SECRETION NYCOMED GMBH (DE) 2008-06-19 WO disclosed