SCHEMBL4574183

SCHEMBL4574183

CCCc1ccc(C(Br)C=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.41
CA2 P00918 1/20 0.40
ACACB O00763 2/20 0.39
LPL P06858 1/20 0.38
LIPG Q9Y5X9 1/20 0.38
MGLL Q99685 1/20 0.38
PLK1 P53350 1/20 0.38
POLB P06746 2/20 0.38
CTDSP1 Q9GZU7 2/20 0.38
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
ACACA Q13085 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17241692 0.89 ALDH1A1 (0.44) THRBCA2PLK1ALDH1A1NPC1
SCHEMBL5709227 0.87 HTR2A (0.47) THRBCA2LPLLIPGALDH1A1
SCHEMBL5141893 0.86 HTR2A (0.50) THRBLPLLIPGMGLLALDH1A1
SCHEMBL15174540 0.86 HTR2A (0.50) THRBLPLLIPGMGLLALDH1A1
SCHEMBL16212189 0.84 MAPK1 (0.45) CA2LPLLIPGMGLLPLK1
SCHEMBL9774407 0.79 LPL (0.43) CA2ACACBLPLLIPGMGLL
SCHEMBL13308116 0.78 ACACB (0.43) THRBCA2ACACBLPLLIPG
SCHEMBL3711064 0.78 ACACB (0.43) THRBCA2ACACBLPLLIPG
SCHEMBL9152292 0.77 LPL (0.45) THRBCA2ACACBLPLLIPG
SCHEMBL6565181 0.77 PTGS1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134036-A1 ALPHA-SUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-α]PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed