SCHEMBL4574889

SCHEMBL4574889

O=CCN1CCN(c2ccc(O)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 2/20 0.54
DRD2 P14416 1/20 0.53
DRD3 P35462 1/20 0.53
ME2 P23368 6/20 0.49
ME1 P48163 6/20 0.49
ME3 Q16798 6/20 0.49
GAA P10253 8/20 0.47
MAPT P10636 4/20 0.47
KDM4E B2RXH2 4/20 0.47
LMNA P02545 1/20 0.47
ALDH1A1 P00352 4/20 0.47
PKM P14618 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
HPGD P15428 1/20 0.46
GFER P55789 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1712413 0.83 CHKA (0.51) DRD4DRD2DRD3GAAMAPT
SCHEMBL1018073 0.82 MAPT (0.61) GAAMAPTKDM4ELMNAALDH1A1
SCHEMBL1412431 0.81 CHRNA7 (0.58) DRD4DRD2DRD3MAPTKDM4E
SCHEMBL17923026 0.81 ALDH1A1 (0.46) DRD4GAAMAPTKDM4EALDH1A1
SCHEMBL23355697 0.80 S1PR1 (0.44) DRD4DRD2DRD3MAPTLMNA
SCHEMBL23780016 0.79 MAPT (0.41) DRD4DRD2DRD3GAAMAPT
SCHEMBL6032280 0.79 CHKA (0.52) DRD4POLB
SCHEMBL27605992 0.79 CHRNA7 (0.38) DRD4DRD2DRD3GAAMAPT
SCHEMBL7041242 0.78 MAPT (0.68) DRD4DRD2DRD3ME2ME1
SCHEMBL3632512 0.77 CTSK (0.60) MAPTLMNAALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014047427-A2 SUBSTITUTED BENZOFURAN, BENZOTHIOPHENE AND INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY (US) 2014-03-27 WO disclosed
WO-2008055959-A1 NOVEL COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS N.V. (BE) 2008-05-15 WO disclosed