SCHEMBL45766

SCHEMBL45766

N=CCN[C@@H](CCCCN)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.49
GSR P00390 1/20 0.44
RNPEP Q9H4A4 1/20 0.43
SLC6A5 Q9Y345 1/20 0.42
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
GGT1 P19440 1/20 0.40
CPB2 Q96IY4 10/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
TLR2 O60603 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676701 1.00 FOLH1 (0.49) FOLH1GSRRNPEPSLC6A5MMP2
Hydrochloric Acid SCHEMBL15923088 0.98 FOLH1 (0.47) FOLH1GSRRNPEPSLC6A5MMP2
Acetic Acid SCHEMBL268741 0.95 FOLH1 (0.45) FOLH1GSRRNPEPSLC6A5MMP2
SCHEMBL232126 0.95 FOLH1 (0.42) FOLH1GSRRNPEPSLC6A5MMP2
SCHEMBL3433410 0.95 FOLH1 (0.42) FOLH1GSRRNPEPSLC6A5MMP2
SCHEMBL27799398 0.95 FOLH1 (0.42) FOLH1GSRRNPEPSLC6A5MMP2
Hydrochloric Acid SCHEMBL15923983 0.93 FOLH1 (0.41) FOLH1GSRRNPEPSLC6A5MMP2
SCHEMBL861645 0.83 FOLH1 (0.49) FOLH1GSRRNPEPSLC6A5MMP2
SCHEMBL861646 0.83 FOLH1 (0.49) FOLH1GSRRNPEPSLC6A5MMP2
SCHEMBL29666181 0.83 FOLH1 (0.49) FOLH1GSRRNPEPSLC6A5MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 348 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088150-B2 Device for disc shunt implantation and peri-shunt injection ALEEVA MEDICAL INC. (US) 2012-01-03 US claimed
US-20090325858-A1 Reduction of Zinc-Induced Neurotoxic Injury By Blockade of Nitric Oxide Synthesis ANDRO DIAGNOSTICS, INC. (US) 2009-12-31 US claimed
US-20090198248-A1 Device for disc shunt implantation and peri-shunt injection YEUNG JEFFREY E 2009-08-06 US claimed
WO-2008080194-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2008-07-10 WO claimed
EP-1534313-A4 OPHTHALMOLOGIC IRRIGATION SOLUTIONS AND METHOD OMEROS CORP (US) 2008-06-25 EP claimed
JP-2007502327-A 2007-02-08 JP claimed
WO-2006084322-A1 TREATMENT METHOD FOR MODIFYING TISSUE PASSIVE ELECTRICAL CONDUCTANCE MCLACHLAN CRAIG STEVEN (AU) 2006-08-17 WO claimed
EP-1631266-A2 A METHOD OF TREATING DEGENERATIVE DISC DISEASE DePuy Spine, Inc. (US) 2006-03-08 EP claimed
WO-2005123130-A2 IMPROVED TREATMENTS OF RHEUMATIC AND ARTHRITIC DISEASES COMPRISING COMBINATIONS OF A 5-LIPOXYGENASE INHIBITOR OSTEOLOGIX A/S (DK) 2005-12-29 WO claimed
WO-2005105065-A2 THIAZOLE-BASED NITRIC OXIDE DONORS FOR TREATING INFLAMMATORY BOWEL DISEASES RENOPHARM LTD. (IL) 2005-11-10 WO claimed
WO-2004084827-A2 REDUCTION OF ZINC-INDUCED NEUROTOXIC INJURY BY BLOCKADE OF NITRIC OXIDE SYNTHESIS NEUROBIOTEX, INC. (US) 2004-10-07 WO claimed
WO-2004010894-A2 OPHTHALMOLOGIC IRRIGATION SOLUTIONS AND METHOD OMEROS CORPORATION (US) 2004-02-05 WO claimed
US-6653350-B1 Modulating interleukin-1 beta levels with n-iminoethyl-lysine G.D. SEARLE & CO. 2003-11-25 US claimed
WO-2003074082-A1 FORMULATIONS AND METHODS OF USING NITRIC OXIDE MIMETICS IN CANCER TREATMENT CELLEGY PHARMACEUTICALS, INC. (CA) 2003-09-12 WO claimed
EP-0966286-B1 ATTENUATION OF OPIOID TOLERANCE BY INHIBITING INDUCIBLE NITRIC OXIDE SYNTHASE PATHWAYS IN THE TREATMENT OF PAIN SEARLE & CO (US) 2003-07-30 EP claimed
US-20020119952-A1 Composition and method of treating arthritis ADVANCED MEDICAL INSTRUMENTS 2002-08-29 US claimed
EP-0866695-A4 COMBINATIONAL THERAPEUTIC METHODS EMPLOYING NITRIC OXIDE SCAVENGERS MEDINOX INC (US) 2001-05-09 EP claimed
EP-0866695-A1 COMBINATIONAL THERAPEUTIC METHODS EMPLOYING NITRIC OXIDE SCAVENGERS Medinox, Inc. (US) 1998-09-30 EP claimed
WO-1997032585-A1 COMBINATIONAL THERAPEUTIC METHODS EMPLOYING NITRIC OXIDE SCAVENGERS AND COMPOSITIONS USEFUL THEREFOR MEDINOX, INC. (US) 1997-09-12 WO claimed
WO-1997018805-A1 COMBINATIONAL THERAPEUTIC METHODS EMPLOYING NITRIC OXIDE SCAVENGERS MEDINOX, INC. (US) 1997-05-29 WO claimed