SCHEMBL457676

SCHEMBL457676

NC(N)c1cc(-c2ccccc2)n[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.55
RAB9A P51151 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.53
TP53 P04637 3/20 0.49
ADORA3 P0DMS8 2/20 0.49
ALOX15 P16050 2/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 2/20 0.44
CYP1A2 P05177 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA2B P29275 1/20 0.44
ADORA1 P30542 1/20 0.44
GSK3B P49841 3/20 0.44
CHEK1 O14757 1/20 0.44
RET P07949 1/20 0.44
PDGFRB P09619 1/20 0.44
PIM1 P11309 1/20 0.44
PDGFRA P16234 1/20 0.44
RPS6KA3 P51812 1/20 0.44
LIMK1 P53667 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2375615 0.81 TP53 (0.63) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL394622 0.80 POLB (0.46) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL15634129 0.78 L3MBTL1 (0.55) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL168659 0.74 POLB (0.61) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL1230353 0.71 RAB9A (1.00) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL12472668 0.71 RAB9A (0.63) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL24566759 0.69 POLB (0.61) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL8795650 0.69 POLB (0.61) POLBRAB9AL3MBTL1TP53ADORA3
SCHEMBL427627 0.69 L3MBTL1 (1.00) POLBRAB9AL3MBTL1TP53LMNA
SCHEMBL9277398 0.69 POLB (0.61) POLBRAB9AL3MBTL1TP53ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015139883-A1 COMPOSITION FOR ALTERING THE COLOR OF KERATIN FIBERS L'OREAL (FR) 2015-09-24 WO disclosed
WO-2013069168-A1 COSMETIC COMPOSITION FOR KERATIN FIBERS L'OREAL (FR) 2013-05-16 WO disclosed
WO-2013069165-A1 COSMETIC COMPOSITION FOR KERATIN FIBERS L'OREAL (FR) 2013-05-16 WO disclosed
WO-2013069166-A1 COSMETIC COMPOSITION FOR KERATIN FIBERS L'OREAL (FR) 2013-05-16 WO disclosed
WO-2012175688-A2 EMULSION DYEING COMPOSITION CONTAINING AN AMINE OR A PHOSPHOLIPID, AT LEAST ONE NONIONIC SURFACTANT AND AT LEAST ONE CARBOXYLIC ACID, AND METHOD OF USING SAME L'OREAL (FR) 2012-12-27 WO disclosed
WO-2012175685-A2 EMULSION DYEING COMPOSITION CONTAINING AN AMINE OR A PHOSPHOLIPID, AT LEAST ONE NONIONIC SURFACTANT AND AT LEAST ONE SILICONE, AND METHOD OF USING SAME L'OREAL (FR) 2012-12-27 WO disclosed
EP-2473235-A1 COMPOSITION COMPRISING AN ACID DYE OF INDIGOID TYPE AND DYEING METHOD L'Oréal (FR) 2012-07-11 EP disclosed
WO-2012032671-A1 COSMETIC COMPOSITION FOR KERATIN FIBERS L'OREAL (FR) 2012-03-15 WO disclosed
EP-2315615-A2 METHODS AND KITS FOR PERMANENTLY COLORING HAIR USING PERSULFATES, PERBORATES OR PERCARBONATES L'Oréal (FR) 2011-05-04 EP disclosed
WO-2011026918-A1 COMPOSITION COMPRISING AN ACID DYE OF INDIGOID TYPE AND DYEING METHOD L'OREAL (FR) 2011-03-10 WO disclosed
EP-2203220-A1 METHODS AND KITS FOR MAINTAINING THE CONDITION OF COLORED HAIR L'Oreal (FR) 2010-07-07 EP disclosed
WO-2010023560-A2 METHODS AND KITS FOR PROVIDING LIFT AND THEN A PERMANENT COLOR TO HAIR L'OREAL (FR) 2010-03-04 WO disclosed
WO-2009098257-A1 COMPOSITION FOR DYEING KERATIN FIBRES COMPRISING AT LEAST ONE CATIONIC DIAMINO-N,N-DIHYDROPYRAZOLONE DERIVATIVE L'OREAL (FR) 2009-08-13 WO disclosed
WO-2009058701-A1 METHODS AND KITS FOR MAINTAINING THE CONDITION OF COLORED HAIR L'OREAL (FR) 2009-05-07 WO disclosed
EP-1868687-A1 AQUEOUS COMPOSITION COMPRISING HYDROGEN PEROXIDE AND INERT PARTICLES L'Oréal (FR) 2007-12-26 EP disclosed
WO-2006106000-A1 AQUEOUS COMPOSITION COMPRISING HYDROGEN PEROXIDE AND INERT PARTICLES L'ORÉAL (FR) 2006-10-12 WO disclosed