SCHEMBL4581583

SCHEMBL4581583

O=C(O)[C@H]1CN(C(=O)NS(=O)(=O)c2ccccc2)CCN1S(=O)(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.50
MMP8 P22894 4/20 0.46
MMP3 P08254 4/20 0.46
STS P08842 1/20 0.44
HCRTR1 O43613 1/20 0.43
HCRTR2 O43614 1/20 0.43
MMP1 P03956 2/20 0.42
MMP7 P09237 2/20 0.42
MMP9 P14780 2/20 0.42
MMP13 P45452 2/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2444870 0.81 MMP1 (0.50) BRD4MMP3MMP1MMP7MMP9
SCHEMBL29178274 0.77 CA12 (0.53) MMP8MMP3MMP9MMP13
SCHEMBL2439382 0.77 MMP1 (0.59) BRD4MMP8MMP3STSMMP1
SCHEMBL2705750 0.75 BRD4 (0.65) BRD4MMP8MMP3HCRTR1HCRTR2
SCHEMBL2705744 0.75 BRD4 (0.65) BRD4MMP8MMP3HCRTR1HCRTR2
SCHEMBL25294154 0.74 KMT2A (0.51) STSMMP1
SCHEMBL5716989 0.74 ALDH1A1 (0.66) BRD4HCRTR1HCRTR2ALDH1A1
SCHEMBL5716988 0.74 ALDH1A1 (0.66) BRD4HCRTR1HCRTR2ALDH1A1
SCHEMBL5717022 0.74 ALDH1A1 (0.66) BRD4HCRTR1HCRTR2ALDH1A1
SCHEMBL25293555 0.73 KMT2A (0.54) STSMMP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2009004-A1 NOVEL PIPERAZINE COMPOUND, AND USE THEREOF AS HCV POLYMERASE INHIBITOR Japan Tobacco, Inc. (JP) 2008-12-31 EP disclosed