SCHEMBL4581815

SCHEMBL4581815

CC(=O)c1ccccc1-c1ccnc(F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.55
ALOX5AP P20292 1/20 0.52
FEN1 P39748 1/20 0.52
CTSA P10619 4/20 0.46
CHEK1 O14757 1/20 0.45
GRM5 P41594 1/20 0.44
PARP10 Q53GL7 1/20 0.43
PARP11 Q9NR21 1/20 0.43
TP53 P04637 1/20 0.40
PDE10A Q9Y233 2/20 0.40
IDO1 P14902 1/20 0.40
ALDH1A1 P00352 1/20 0.40
DPP4 P27487 1/20 0.39
ELOVL1 Q9BW60 1/20 0.39
DAPK3 O43293 1/20 0.39
JAK2 O60674 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
PAK4 O96013 1/20 0.39
ABL1 P00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6215832 0.83 PARP10 (0.39) KDM4CALOX5APFEN1CTSAGRM5
SCHEMBL2559099 0.81 KDM4C (0.62) KDM4CALOX5APFEN1CTSACHEK1
SCHEMBL1515697 0.79 ALOX5AP (0.59) KDM4CALOX5APFEN1CTSACHEK1
SCHEMBL9208056 0.76 ALDH1A1 (0.58) KDM4CALOX5APFEN1CHEK1TP53
SCHEMBL29466481 0.76 HTT (0.57) KDM4CALOX5APFEN1CTSACHEK1
SCHEMBL1515901 0.76 HTT (0.57) KDM4CALOX5APFEN1CTSACHEK1
SCHEMBL11781294 0.75 KDM4C (0.53) KDM4CALOX5APFEN1CTSACHEK1
SCHEMBL28493426 0.75 ALDH1A1 (0.47) ALOX5APFEN1GRM5IDO1ALDH1A1
SCHEMBL4745781 0.75 CTSA (0.51) KDM4CALOX5APFEN1CTSACHEK1
SCHEMBL29354773 0.74 ADORA2B (0.40) PARP10PARP11PDE10AIDO1MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899370-A1 A CRYSTAL STRUCTURE AND USES THEREOF MONASH UNIVERSITY (AU) 2008-03-19 EP disclosed
WO-2006119542-A1 A CRYSTAL STRUCTURE AND USES THEREOF CYTOPIA RESEARCH PTY LTD (AU) 2006-11-16 WO disclosed