SCHEMBL4582601

SCHEMBL4582601

COC(=O)Oc1cc2c(s1)CCN(C)CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
HPGD P15428 2/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
ABCB11 O95342 1/20 0.38
CHRM2 P08172 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
AR P10275 1/20 0.38
OPRM1 P35372 1/20 0.38
P2RY12 Q9H244 1/20 0.38
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
POLB P06746 2/20 0.36
PKM P14618 1/20 0.36
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.34
SLC6A4 P31645 1/20 0.34
HDAC6 Q9UBN7 2/20 0.33
MAPT P10636 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4431441 0.92 WDR91 (0.41) ALDH1A1HPGDMAOAMAOBSLC6A4
SCHEMBL4433208 0.85 ABCB11 (0.36) ALDH1A1HPGDTP53MAPK1ABCB11
SCHEMBL4440893 0.80 CYP3A4 (0.31) MAOAMAOBSLC6A4DRD1DRD5
SCHEMBL4435195 0.79 PNMT (0.42) ALDH1A1HPGDTP53MAPK1ABCB11
SCHEMBL4431719 0.78 SLC6A2 (0.31) ABCB11CHRM2ADORA3AROPRM1
SCHEMBL4440822 0.77 PRMT5 (0.38) ALDH1A1HPGDMAPK1ABCB11CHRM2
SCHEMBL19933106 0.77 MEN1 (0.39) ALDH1A1ABCB11CHRM2ADORA3AR
SCHEMBL4440903 0.77 PARP1 (0.41) ALDH1A1HPGDABCB11CHRM2ADORA3
SCHEMBL4433993 0.77 PARP1 (0.41) ALDH1A1HPGDMAOAMAOBSLC6A4
SCHEMBL16869983 0.77 ABCB11 (0.49) ALDH1A1HPGDABCB11CHRM2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132193-B1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INT (DE) 2012-10-24 EP disclosed
EP-1975165-A1 Substituted pyrrolidinamides, their production and utilisation as medicine Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2008-10-01 EP disclosed