SCHEMBL4582735

SCHEMBL4582735

O=C(O)c1sc(-c2ccnc3c2ccn3S(=O)(=O)c2ccccc2)c(Br)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.41
PIK3C3 Q8NEB9 3/20 0.37
HTR6 P50406 6/20 0.35
ENPP3 O14638 2/20 0.35
ENPP1 P22413 2/20 0.35
MET P08581 1/20 0.34
HDAC3 O15379 3/20 0.34
HDAC4 P56524 3/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC7 Q8WUI4 3/20 0.34
HDAC2 Q92769 3/20 0.34
HDAC10 Q969S8 3/20 0.34
HDAC11 Q96DB2 3/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC9 Q9UKV0 3/20 0.34
HDAC5 Q9UQL6 3/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4612732 0.90 PIK3C3 (0.42) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL4582645 0.89 CYP2C19 (0.42) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL4582484 0.86 CYP2C19 (0.39) CYP2C19PIK3C3HTR6DRD2HTR2A
SCHEMBL4584711 0.81 PIK3C3 (0.40) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL8242820 0.81 PIK3C3 (0.40) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL4591926 0.76 AKT1 (0.43) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL4633196 0.75 CYP2C19 (0.46) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL27848203 0.74 CYP2C19 (0.45) CYP2C19PIK3C3HTR6ENPP3ENPP1
SCHEMBL4582702 0.74 HTR6 (0.36) PIK3C3HTR6
SCHEMBL16052009 0.73 CYP2C19 (0.52) CYP2C19HTR6METDRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed