SCHEMBL458280

SCHEMBL458280

NC(=O)OC(CC(F)(F)F)c1cc(NC2CCCC2)nn2c(I)cnc12

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 7/20 0.43
TTK P33981 4/20 0.35
STAT3 P40763 1/20 0.32
CDK2 P24941 8/20 0.32
CCNA2 P20248 2/20 0.32
CCNA1 P78396 2/20 0.32
CCNE1 P24864 6/20 0.32
FLT3 P36888 6/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL458281 0.72 TYK2 (0.40) TYK2TTKCDK2CCNE1FLT3
SCHEMBL455869 0.71 TYK2 (0.41) TYK2TTKCDK2CCNE1FLT3
SCHEMBL470186 0.70 TYK2 (0.45) TYK2TTKCDK2CCNE1FLT3
SCHEMBL21571914 0.61 TYK2 (1.00) TYK2TTKSTAT3CDK2CCNE1
SCHEMBL458935 0.56 TTK (0.41) TTK
SCHEMBL28629637 0.54 CYP17A1 (0.31)
SCHEMBL22421804 0.54 TYK2 (0.77) TYK2STAT3CDK2CCNE1FLT3
SCHEMBL19516750 0.54 MEN1 (0.42)
SCHEMBL3033387 0.53 PIM1 (0.60) CDK2FLT3
SCHEMBL3033386 0.53 PIM1 (0.60) CDK2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-B1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-01-13 EP disclosed
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed