SCHEMBL455869

SCHEMBL455869

O=C(O)N(CCC(F)(F)F)c1cc(NC2CCCC2)nn2c(I)cnc12

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 4/20 0.41
TTK P33981 4/20 0.36
HCAR3 P49019 2/20 0.33
MKNK1 Q9BUB5 1/20 0.32
MAPK14 Q16539 1/20 0.32
IRAK4 Q9NWZ3 3/20 0.31
CSNK2B P67870 1/20 0.31
IKBKB O14920 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
FLT3 P36888 1/20 0.31
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17425401 0.88 TYK2 (0.37) TYK2TTKIRAK4
SCHEMBL456788 0.82 CCNE1 (0.35) TYK2TTKHCAR3MAPK14IRAK4
SCHEMBL17416356 0.78 TTK (0.59) TTK
SCHEMBL470186 0.75 TYK2 (0.45) TYK2TTKCCNE1CDK2FLT3
SCHEMBL458281 0.75 TYK2 (0.40) TYK2TTKCCNE1CDK2FLT3
SCHEMBL17425406 0.71 IRAK4 (0.34) TYK2TTKIRAK4CCNE1CDK2
SCHEMBL458280 0.71 TYK2 (0.43) TYK2TTKCCNE1CDK2FLT3
SCHEMBL17425402 0.69 TTK (0.56) TTK
SCHEMBL139927 0.69 TTK (0.47) TTKMAPK14
SCHEMBL12986323 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-B1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER IP GMBH (DE) 2016-01-13 EP disclosed
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed