SCHEMBL4582983

SCHEMBL4582983

Nc1cc(-c2cn(S(=O)(=O)c3ccccc3)c3ncccc23)c(-c2cccnc2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.43
CDK8 P49336 1/20 0.43
HTR6 P50406 6/20 0.41
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
CYP2C19 P33261 1/20 0.38
DRD2 P14416 2/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38
ELANE P08246 1/20 0.37
CKS1B P61024 2/20 0.36
SKP2 Q13309 2/20 0.36
PDPK1 O15530 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4583354 0.79 HTR6 (0.42) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL4584006 0.77 HTR6 (0.41) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL13332928 0.74 HTR6 (0.50) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL29605131 0.73 HTR6 (0.46) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL1044724 0.73 CDK2 (0.47) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL2529105 0.73 HTR6 (0.51) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL8233323 0.72 HTR6 (0.39) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL29606686 0.71 HTR6 (0.51) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL17165465 0.71 CCNC (0.52) CCNCCDK8HTR6CCNE1CDK2
SCHEMBL1049986 0.71 CYP2C19 (0.49) CCNCCDK8HTR6CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed