SCHEMBL4584006

SCHEMBL4584006

O=C(O)Nc1cc(-c2cn(S(=O)(=O)c3ccccc3)c3ncccc23)c(-c2ccccc2)s1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 10/20 0.41
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
CYP2C19 P33261 1/20 0.38
PIK3C3 Q8NEB9 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8233323 0.89 HTR6 (0.39) HTR6CCNCCDK8CCNE1CDK2
SCHEMBL4583354 0.85 HTR6 (0.42) HTR6CCNCCDK8CCNE1CDK2
SCHEMBL4584452 0.82 HTR6 (0.44) HTR6CCNCCDK8CCNE1CDK2
SCHEMBL8241863 0.80 ELANE (0.38) HTR6CCNCCDK8CCNE1CDK2
SCHEMBL4583381 0.79 PTPRB (0.41) HTR6CDK2
SCHEMBL4582983 0.77 CCNC (0.43) HTR6CCNCCDK8CCNE1CDK2
SCHEMBL4476225 0.76 L3MBTL1 (0.45) PTGDR2L3MBTL1
SCHEMBL4591926 0.75 AKT1 (0.43) HTR6CYP2C19PIK3C3L3MBTL1
SCHEMBL8944259 0.72 L3MBTL1 (0.67) HTR6CCNCCDK8PTGDR2CYP2C19
SCHEMBL17165375 0.72 HTR6 (0.45) HTR6CCNCCDK8CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed