SCHEMBL4583354

SCHEMBL4583354

O=C(O)c1cc(-c2cn(S(=O)(=O)c3ccccc3)c3ncccc23)c(-c2ccccc2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 7/20 0.42
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
CYP2C19 P33261 1/20 0.40
CDK2 P24941 3/20 0.39
CCNE1 P24864 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
MAPK14 Q16539 1/20 0.38
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PLK4 O00444 1/20 0.37
AURKA O14965 1/20 0.37
DAPK3 O43293 1/20 0.37
CHEK2 O96017 1/20 0.37
CDK1 P06493 1/20 0.37
PIM1 P11309 1/20 0.37
PRKACA P17612 1/20 0.37
MAPK9 P45984 1/20 0.37
CSNK1D P48730 1/20 0.37
GSK3A P49840 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4584006 0.85 HTR6 (0.41) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL8233323 0.80 HTR6 (0.39) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL4582983 0.79 CCNC (0.43) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL3355302 0.76 HTR6 (0.45) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL17165465 0.73 CCNC (0.52) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL2529105 0.73 HTR6 (0.51) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL1049986 0.73 CYP2C19 (0.49) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL4584452 0.73 HTR6 (0.44) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL1584951 0.72 HTR6 (0.47) HTR6CCNCCDK8CYP2C19CDK2
SCHEMBL8944259 0.72 L3MBTL1 (0.67) HTR6CCNCCDK8CYP2C19PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed