SCHEMBL4583765

SCHEMBL4583765

O=C(O)NCC(Cc1ccccc1)NC(=O)c1coc(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 5/20 0.47
KLK7 P49862 1/20 0.43
PIN1 Q13526 3/20 0.43
CTSL P07711 4/20 0.42
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
RPS6KA4 O75676 1/20 0.40
PRKACA P17612 1/20 0.40
MAPK1 P28482 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
IRAK1 P51617 1/20 0.40
PRKX P51817 1/20 0.40
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3509771 0.77 CTRB1 (0.42) CTRB1PIN1CTSLTP53HPGD
SCHEMBL11884009 0.76 CTRB1 (0.49) CTRB1MAPK1MMENPC1RAB9A
SCHEMBL4581842 0.75 ALDH1A1 (0.40) CTRB1KLK7CTSLALDH1A1LMNA
SCHEMBL3506437 0.75 ALDH1A1 (0.48) CTRB1PIN1CTSLALDH1A1LMNA
SCHEMBL3506435 0.75 ALDH1A1 (0.48) CTRB1PIN1CTSLALDH1A1LMNA
SCHEMBL3511843 0.75 ALDH1A1 (0.48) CTRB1PIN1CTSLALDH1A1LMNA
SCHEMBL3509337 0.74 AKT1 (0.48) CTRB1PIN1ALDH1A1LMNAGSK3B
SCHEMBL3505511 0.73 KMT2A (0.48) CTRB1PIN1ALDH1A1LMNAHPGD
SCHEMBL3507223 0.72 CTRB1 (0.42) CTRB1PIN1CTSLALDH1A1HPGD
SCHEMBL3510049 0.72 KMT2A (0.41) CTRB1PIN1CTSLALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968568-A2 INHIBITORS OF Akt ACTIVITY SmithKline Beecham Corporation (US) 2008-09-17 EP disclosed
WO-2007076423-A2 INHIBITORS OF Akt ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-07-05 WO disclosed