SCHEMBL45838

SCHEMBL45838

COc1ccc(O[Si](C)(C)C(C)(C)C)c(C(C)(O)c2nc3ccc(OC)cc3s2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 5/20 0.47
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 2/20 0.43
PDK1 Q15118 1/20 0.42
MAPT P10636 4/20 0.42
TSHR P16473 2/20 0.42
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
HTT P42858 1/20 0.40
DYRK1A Q13627 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
CASP1 P29466 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30731274 0.76 CYP1A2 (0.58) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL31285 0.75 HSD17B1 (0.51) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL799881 0.73 CYP1A2 (0.61) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL30663 0.72 GAA (0.50) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL30666 0.72 HSD17B1 (0.59) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL19435592 0.70 CYP1A2 (0.59) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL21652231 0.69 CYP1A2 (0.55) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL2055276 0.69 CA12 (0.46) CYP1A2CYP3A4CYP2C19PDK1MAPT
SCHEMBL13640332 0.68 CA12 (0.59) CYP1A2CYP3A4CYP2C19MAPTMEN1
SCHEMBL31558330 0.68 TDP1 (0.56) CYP1A2CYP3A4CYP2C19PDK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed