SCHEMBL4585160

SCHEMBL4585160

C/C(=C\CCl)CCc1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 3/20 0.51
MMP12 P39900 2/20 0.46
LSS P48449 1/20 0.43
NAAA Q02083 1/20 0.42
ALDH1A1 P00352 1/20 0.42
FFAR4 Q5NUL3 1/20 0.41
KCNH2 Q12809 1/20 0.40
TRPV1 Q8NER1 2/20 0.40
HDAC2 Q92769 2/20 0.40
CES1 P23141 2/20 0.39
HDAC1 Q13547 1/20 0.39
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2813151 0.85 FFAR1 (0.53) FFAR1MMP12LSSNAAAALDH1A1
SCHEMBL5808516 0.82 FFAR1 (0.58) FFAR1MMP12NAAAALDH1A1FFAR4
SCHEMBL14596301 0.80 ICMT (0.46) FFAR1MMP12LSSNAAAALDH1A1
SCHEMBL29408009 0.74 ALDH1A1 (0.55) FFAR1ALDH1A1TRPV1HDAC2HDAC1
SCHEMBL29572084 0.73 ALDH1A1 (0.53) FFAR1LSSALDH1A1TRPV1HDAC2
SCHEMBL21486330 0.73 ALDH1A1 (0.53) FFAR1LSSALDH1A1TRPV1HDAC2
SCHEMBL8260837 0.73 ALDH1A1 (0.77) FFAR1MMP12NAAAALDH1A1FFAR4
SCHEMBL29105881 0.73 ALDH1A1 (0.53) FFAR1LSSALDH1A1TRPV1HDAC2
SCHEMBL29098167 0.72 FFAR1 (0.58) FFAR1MMP12NAAAALDH1A1FFAR4
SCHEMBL9637227 0.72 FFAR1 (0.48) FFAR1MMP12LSSKCNH2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613585-A4 COMPOUNDS AND METHODS FOR USE IN TREATING NEOPLASIA AND CANCER BASED UPON INHIBITORS OF ISOPRENYLCYSTEINE METHYLTRANSFERASE PURDUE RESEARCH FOUNDATION (US) 2008-07-23 EP disclosed
EP-1613585-A2 COMPOUNDS AND METHODS FOR USE IN TREATING NEOPLASIA AND CANCER BASED UPON INHIBITORS OF ISOPRENYLCYSTEINE METHYLTRANSFERASE PURDUE RESEARCH FOUNDATION (US) 2006-01-11 EP disclosed
WO-2004087064-A2 COMPOUNDS AND METHODS FOR USE IN TREATING NEOPLASIA AND CANCER BASED UPON INHIBITORS OF ISOPRENYLCYSTEINE METHYLTRANSFERASE PURDUE RESEARCH FOUNDATION (US) 2004-10-14 WO disclosed