SCHEMBL4585691

SCHEMBL4585691

O=C1N=C(Nc2c(Cl)cccc2Cl)S/C1=C\c1ccc2ncc(C(=O)O)c(Cl)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CISD1 Q9NZ45 1/20 0.41
EGFR P00533 4/20 0.36
SRC P12931 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NSD2 O96028 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
APEX1 P27695 1/20 0.34
RECQL P46063 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ENPP2 Q13822 1/20 0.34
CSF1R P07333 2/20 0.34
DYRK3 O43781 1/20 0.34
CSNK1E P49674 1/20 0.34
CLK1 P49759 1/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4585695 1.00 CISD1 (0.41) CISD1EGFRSRCMEN1KMT2A
SCHEMBL4586074 0.88 CISD1 (0.40) CISD1EGFRSRCMEN1KMT2A
SCHEMBL4586069 0.88 CISD1 (0.40) CISD1EGFRSRCMEN1KMT2A
SCHEMBL2984471 0.87 MAPT (0.44) CISD1SRCMEN1KMT2AKDM4E
SCHEMBL4586095 0.87 MAPT (0.44) CISD1SRCMEN1KMT2AKDM4E
SCHEMBL4585835 0.84 MEN1 (0.47) CISD1MEN1KMT2AKDM4EPOLB
SCHEMBL4585846 0.84 MEN1 (0.47) CISD1MEN1KMT2AKDM4EPOLB
SCHEMBL4586124 0.84 ENPP2 (0.45) CISD1MEN1KMT2AENPP2CSF1R
Trifluoroacetic Acid SCHEMBL2985105 0.84 CISD1 (0.39) CISD1EGFRSRCMEN1KMT2A
Trifluoroacetic Acid SCHEMBL2985114 0.84 CISD1 (0.39) CISD1EGFRSRCMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP disclosed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP disclosed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO disclosed