SCHEMBL4587397

SCHEMBL4587397

CCc1nc2ccc(/C=C3\SC(Nc4cc(NC(=O)C(C)C)ccc4Cl)=NC3=O)cc2cc1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.38
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
CISD1 Q9NZ45 1/20 0.34
IGF1R P08069 1/20 0.33
HDAC4 P56524 2/20 0.32
ENPP2 Q13822 1/20 0.32
NPC1 O15118 4/20 0.31
RAB9A P51151 4/20 0.31
KDM4E B2RXH2 3/20 0.31
SMN1; SMN2 Q16637 3/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
CASP3 P42574 2/20 0.31
SENP7 Q9BQF6 2/20 0.31
NR2E3 Q9Y5X4 1/20 0.31
MCHR1 Q99705 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
RECQL P46063 1/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4587403 1.00 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ACISD1IGF1R
Trifluoroacetic Acid SCHEMBL2995754 0.96 ALDH1A1 (0.35) ALDH1A1MEN1KMT2ACISD1IGF1R
Trifluoroacetic Acid SCHEMBL2995750 0.96 ALDH1A1 (0.35) ALDH1A1MEN1KMT2ACISD1IGF1R
SCHEMBL4586161 0.87 PTGDR2 (0.34) CISD1HDAC4ENPP2PTGDR2NR2E3
SCHEMBL4586168 0.87 PTGDR2 (0.34) CISD1HDAC4ENPP2PTGDR2NR2E3
SCHEMBL4586480 0.84 IGF1R (0.37) ALDH1A1MEN1KMT2ACISD1IGF1R
Trifluoroacetic Acid SCHEMBL2991042 0.83 EGFR (0.33) CISD1HDAC4PTGDR2NR2E3MCHR1
Trifluoroacetic Acid SCHEMBL2991046 0.83 EGFR (0.33) CISD1HDAC4PTGDR2NR2E3MCHR1
SCHEMBL2988362 0.83 FABP3 (0.39) ALDH1A1MEN1KMT2ACISD1IGF1R
SCHEMBL2996479 0.81 DYRK3 (0.42) ALDH1A1MEN1KMT2ACISD1IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879563-A4 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2008-07-16 EP claimed
EP-1879563-A2 NOVEL CHEMICAL COMPOUNDS Smithkline Beecham Corporation (US) 2008-01-23 EP claimed
WO-2006132739-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-14 WO claimed